A Development of Chimeric VEGFR2 TK Inhibitor Based on Two Ligand Conformers from PDB: 1Y6A Complex - Medicinal Chemistry Consequences of a TKs Analysis Lucia Lintnerová, a Melissa García-Caballero, b Fridrich Gregáň, c Milan Melicherčík, c Ana R. Quesada, b Juraj Dobiaš, a Ján Lác, d Marta Sališová, a and Andrej Boháč, a,d* a Comenius University, Faculty of Natural Sciences, Department of Organic Chemistry, Mlynská dolina 842 15, Bratislava, Slovakia, [email protected], phone: +421260296409, fax: +421260296337 b Departamento de Biología Molecular y Bioquímica, Facultad de Ciencias, Universidad de Málaga, Campus de Teatinos, 29071-Málaga, Spain. Tel. 34(9)52137128, Fax. 34(9)52132000, [email protected] c Matej Bel University, Faculty of Natural Sciences, Department of Chemistry Tajovského 40, 974 01 Banská Bystrica, Slovakia, [email protected], [email protected] d Biomagi, Inc., Mamateyova 26, 851 04 Bratislava, Slovakia, phone: +421902522144 1